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(R)-(-)-JQ1 Enantiomer
CAS No. 1268524-71-5
(R)-(-)-JQ1 Enantiomer ( —— )
产品货号. M11127 CAS No. 1268524-71-5
(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1, (+)-JQ-1 is a potent, specific BET bromodomain BRD4 inhibitor.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 2MG | ￥494 | 有现货 |
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| 5MG | ￥948 | 有现货 |
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| 10MG | ￥1596 | 有现货 |
|
| 25MG | ￥3216 | 有现货 |
|
| 50MG | ￥5014 | 有现货 |
|
| 100MG | ￥7120 | 有现货 |
|
| 200MG | 获取报价 | 有现货 |
|
| 500MG | 获取报价 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称(R)-(-)-JQ1 Enantiomer
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1, (+)-JQ-1 is a potent, specific BET bromodomain BRD4 inhibitor.
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产品描述(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1, (+)-JQ-1 is a potent, specific BET bromodomain BRD4 inhibitor, but (-)-JQ1 has no activity.
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同义词——
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通路Chromatin/Epigenetic
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靶点Bromodomain
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受体Bromodomain
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研究领域Cancer
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适应症——
化学信息
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CAS Number1268524-71-5
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分子量456.99
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分子式C23H25ClN4O2S
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纯度>98% (HPLC)
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溶解度10 mM in DMSO
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SMILESCC1=C(SC2=C1C(=NC(C3=NN=C(N32)C)CC(=O)OC(C)(C)C)C4=CC=C(C=C4)Cl)C
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化学全称6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-trimethyl-, 1,1-dimethylethyl ester, (6R)-
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Filippakopoulos P, et al. Nature. 2010 Dec 23;468(7327):1067-73.
产品手册
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